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Atypical nicotinic agonist bound conformations conferring subtype selectivity

The nicotinic acetylcholine (ACh) receptor (nAChR) plays a crucial role in excitatory neurotransmission and is an important target for drugs and insecticides. Diverse nAChR subtypes with various subunit combinations confer differential selectivity for nicotinic drugs. We investigated the subtype sel...

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Detalles Bibliográficos
Main Authors: Tomizawa, Motohiro, Maltby, David, Talley, Todd T., Durkin, Kathleen A., Medzihradszky, Katalin F., Burlingame, Alma L., Taylor, Palmer, Casida, John E.
Formato: Artigo
Idioma:Inglês
Publicado: National Academy of Sciences 2008
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC2234212/
https://ncbi.nlm.nih.gov/pubmed/18230720
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0711724105
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