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Long-acting κ Opioid Antagonists Disrupt Receptor Signaling and Produce Noncompetitive Effects by Activating c-Jun N-terminal Kinase

Norbinaltorphimine (NorBNI), guanidinonaltrindole, and atrans-(3R,4R)-dimethyl-4-(3-hydroxyphenyl) piperidine (JDTic) are selective κ opioid receptor (KOR) antagonists having very long durations of action in vivo despite binding non-covalently in vitro and having only moderately high affinities. Con...

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Bibliografske podrobnosti
Main Authors: Bruchas, Michael R., Yang, Tao, Schreiber, Selena, DeFino, Mia, Kwan, Steven C., Li, Shuang, Chavkin, Charles
Format: Artigo
Jezik:Inglês
Izdano: 2007
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC2096775/
https://ncbi.nlm.nih.gov/pubmed/17702750
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M705540200
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