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Hot-spot mimicry of a cytokine receptor by a small molecule

Protein–protein complexes remain enticing, but extremely challenging, targets for small-molecule drug discovery. In a rare example described earlier, a high-affinity small molecule, SP4206 (K(d) ≈ 70 nM), was found to block binding of the IL-2α receptor (IL-2Rα) to IL-2 (K(d) ≈ 10 nM). Recently, the...

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Detalhes bibliográficos
Main Authors: Thanos, Christopher D., DeLano, Warren L., Wells, James A.
Formato: Artigo
Idioma:Inglês
Publicado em: National Academy of Sciences 2006
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1592646/
https://ncbi.nlm.nih.gov/pubmed/17032757
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0607058103
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