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Structural basis for antibiotic recognition by the TipA class of multidrug-resistance transcriptional regulators

The TipAL protein, a bacterial transcriptional regulator of the MerR family, is activated by numerous cyclic thiopeptide antibiotics. Its C-terminal drug-binding domain, TipAS, defines a subfamily of broadly distributed bacterial proteins including Mta, a central regulator of multidrug resistance in...

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Detalles Bibliográficos
Main Authors: Kahmann, Jan D., Sass, Hans-Jürgen, Allan, Martin G., Seto, Haruo, Thompson, Charles J., Grzesiek, Stephan
Formato: Artigo
Idioma:Inglês
Publicado: Oxford University Press 2003
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC154473/
https://ncbi.nlm.nih.gov/pubmed/12682015
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/emboj/cdg181
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