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Structures of eukaryotic ribonucleotide reductase I define gemcitabine diphosphate binding and subunit assembly

Ribonucleotide reductase (RNR) catalyzes the conversion of nucleoside diphosphates to deoxynucleoside diphosphates. Crucial for rapidly dividing cells, RNR is a target for cancer therapy. In eukaryotes, RNR comprises a heterooligomer of α(2) and β(2) subunits. Rnr1, the α subunit, contains regulator...

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Autors principals: Xu, Hai, Faber, Catherine, Uchiki, Tomoaki, Racca, Joseph, Dealwis, Chris
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2006
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1389703/
https://ncbi.nlm.nih.gov/pubmed/16537480
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0600440103
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