Design and Characterization of a Novel Fluorinated Magnetic Resonance Imaging Agent for Functional Analysis of Bile Acid Transporter Activity

Por Vivian, Diana, Cheng, Kunrong, Khurana, Sandeep, Xu, Su, Whiterock, Valerie, Witter, Drew, Lentz, Kimberley A., Santone, Kenneth S., Raufman, Jean-Pierre, Polli, James E.
Publicado em 2013

Preclinical Characterization of BMS-791325, an Allosteric Inhibitor of Hepatitis C Virus NS5B Polymerase

Por Lemm, Julie A., Liu, Mengping, Gentles, Robert G., Ding, Min, Voss, Stacey, Pelosi, Lenore A., Wang, Ying-Kai, Rigat, Karen L., Mosure, Kathleen W., Bender, John A., Knipe, Jay O., Colonno, Richard, Meanwell, Nicholas A., Kadow, John F., Santone, Kenneth S., Roberts, Susan B., Gao, Min
Publicado em 2014

Development of 1H-Pyrazolo[3,4-b]pyridines as Metabotropic Glutamate Receptor 5 Positive Allosteric Modulators

Por Hill, Matthew D., Fang, Haiquan, Brown, Jeffrey M., Molski, Thaddeus, Easton, Amy, Han, Xiaojun, Miller, Regina, Hill-Drzewi, Melissa, Gallagher, Lizbeth, Matchett, Michele, Gulianello, Michael, Balakrishnan, Anand, Bertekap, Robert L., Santone, Kenneth S., Whiterock, Valerie J., Zhuo, Xiaoliang, Bronson, Joanne J., Macor, John E., Degnan, Andrew P.
Publicado no ACS Med Chem Lett (2016)

Discovery and Preclinical Evaluation of BMS-955829, a Potent Positive Allosteric Modulator of mGluR5

Por Yang, Fukang, Snyder, Lawrence B., Balakrishnan, Anand, Brown, Jeffrey M., Sivarao, Digavalli V., Easton, Amy, Fernandes, Alda, Gulianello, Michael, Hanumegowda, Umesh M., Huang, Hong, Huang, Yanling, Jones, Kelli M., Li, Yu-Wen, Matchett, Michele, Mattson, Gail, Miller, Regina, Santone, Kenneth S., Senapati, Arun, Shields, Eric E., Simutis, Frank J., Westphal, Ryan, Whiterock, Valerie J., Bronson, Joanne J., Macor, John E., Degnan, Andrew P.
Publicado no ACS Med Chem Lett (2016)

Discovery of BMS-955176, a Second Generation HIV-1 Maturation Inhibitor with Broad Spectrum Antiviral Activity

Por Regueiro-Ren, Alicia, Liu, Zheng, Chen, Yan, Sin, Ny, Sit, Sing-Yuen, Swidorski, Jacob J., Chen, Jie, Venables, Brian L., Zhu, Juliang, Nowicka-Sans, Beata, Protack, Tricia, Lin, Zeyu, Terry, Brian, Samanta, Himadri, Zhang, Sharon, Li, Zhufang, Beno, Brett R., Huang, Xiaohua S., Rahematpura, Sandhya, Parker, Dawn D., Haskell, Roy, Jenkins, Susan, Santone, Kenneth S., Cockett, Mark I., Krystal, Mark, Meanwell, Nicholas A., Hanumegowda, Umesh, Dicker, Ira B.
Publicado no ACS Med Chem Lett (2016)

Inhibition of AAK1 Kinase as a Novel Therapeutic Approach to Treat Neuropathic Pain

Por Kostich, Walter, Hamman, Brian D., Li, Yu-Wen, Naidu, Sreenivasulu, Dandapani, Kumaran, Feng, Jianlin, Easton, Amy, Bourin, Clotilde, Baker, Kevin, Allen, Jason, Savelieva, Katerina, Louis, Justin V., Dokania, Manoj, Elavazhagan, Saravanan, Vattikundala, Pradeep, Sharma, Vivek, Das, Manish Lal, Shankar, Ganesh, Kumar, Anoop, Holenarsipur, Vinay K., Gulianello, Michael, Molski, Ted, Brown, Jeffrey M., Lewis, Martin, Huang, Yanling, Lu, Yifeng, Pieschl, Rick, O’Malley, Kevin, Lippy, Jonathan, Nouraldeen, Amr, Lanthorn, Thomas H., Ye, Guilan, Wilson, Alan, Balakrishnan, Anand, Denton, Rex, Grace, James E., Lentz, Kimberley A., Santone, Kenneth S., Bi, Yingzhi, Main, Alan, Swaffield, Jon, Carson, Ken, Mandlekar, Sandhya, Vikramadithyan, Reeba K., Nara, Susheel J., Dzierba, Carolyn, Bronson, Joanne, Macor, John E., Zaczek, Robert, Westphal, Ryan, Kiss, Laszlo, Bristow, Linda, Conway, Charles M., Zambrowicz, Brian, Albright, Charles F.
Publicado no J Pharmacol Exp Ther (2016)