Discovery of New 1,1′-Biphenyl-4-sulfonamides as Selective Subnanomolar Human Carbonic Anhydrase II Inhibitors

по La Regina, Giuseppe, Puxeddu, Michela, Nalli, Marianna, Vullo, Daniela, Gratteri, Paola, Supuran, Claudiu Trandafir, Nocentini, Alessio, Silvestri, Romano
Опубликовано в: ACS Med Chem Lett (2019)

Modeling Epac1 interactions with the allosteric inhibitor AM-001 by co-solvent molecular dynamics

по Bufano, Marianna, Laudette, Marion, Blondeau, Jean-Paul, Lezoualc’h, Frank, Nalli, Marianna, Silvestri, Romano, Brancale, Andrea, Coluccia, Antonio
Опубликовано в: J Comput Aided Mol Des (2020)

Discovery of Kynurenines Containing Oligopeptides as Potent Opioid Receptor Agonists

по Szűcs, Edina, Stefanucci, Azzurra, Dimmito, Marilisa Pia, Zádor, Ferenc, Pieretti, Stefano, Zengin, Gokhan, Vécsei, László, Benyhe, Sándor, Nalli, Marianna, Mollica, Adriano
Опубликовано в: Biomolecules (2020)

Discovery of Zika Virus NS2B/NS3 Inhibitors That Prevent Mice from Life-Threatening Infection and Brain Damage

по Coluccia, Antonio, Puxeddu, Michela, Nalli, Marianna, Wei, Chih-Ku, Wu, Yu-Hsuan, Mastrangelo, Eloise, Elamin, Tasneem, Tarantino, Delia, Bugert, Joachim Jakob, Schreiner, Benno, Nolte, Juliane, Schwarze, Frank, La Regina, Giuseppe, Lee, Jin-Ching, Silvestri, Romano
Опубликовано в: ACS Med Chem Lett (2020)

Drug Design and Synthesis of First in Class PDZ1 Targeting NHERF1 Inhibitors as Anticancer Agents

по Coluccia, Antonio, La Regina, Giuseppe, Naccarato, Valentina, Nalli, Marianna, Orlando, Viviana, Biagioni, Stefano, De Angelis, Maria Laura, Baiocchi, Marta, Gautier, Candice, Gianni, Stefano, Di Pastena, Fiorella, Di Magno, Laura, Canettieri, Gianluca, Coluccia, Addolorata Maria Luce, Silvestri, Romano
Опубликовано в: ACS Med Chem Lett (2019)

3-Aroyl-1,4-diarylpyrroles Inhibit Chronic Myeloid Leukemia Cell Growth through an Interaction with Tubulin

по La Regina, Giuseppe, Bai, Ruoli, Coluccia, Antonio, Famiglini, Valeria, Passacantilli, Sara, Naccarato, Valentina, Ortar, Giorgio, Mazzoccoli, Carmela, Ruggieri, Vitalba, Agriesti, Francesca, Piccoli, Claudia, Tataranni, Tiziana, Nalli, Marianna, Brancale, Andrea, Vultaggio, Stefania, Mercurio, Ciro, Varasi, Mario, Saponaro, Concetta, Sergio, Sara, Maffia, Michele, Coluccia, Addolorata Maria Luce, Hamel, Ernest, Silvestri, Romano
Опубликовано в: ACS Med Chem Lett (2017)

New Pyrrole Derivatives with Potent Tubulin Polymerization Inhibiting Activity As Anticancer Agents Including Hedgehog-Dependent Cancer

по La Regina, Giuseppe, Bai, Ruoli, Coluccia, Antonio, Famiglini, Valeria, Pelliccia, Sveva, Passacantilli, Sara, Mazzoccoli, Carmela, Ruggieri, Vitalba, Sisinni, Lorenza, Bolognesi, Alessio, Rensen, Whilelmina Maria, Miele, Andrea, Nalli, Marianna, Alfonsi, Romina, Di Marcotullio, Lucia, Gulino, Alberto, Brancale, Andrea, Novellino, Ettore, Dondio, Giulio, Vultaggio, Stefania, Varasi, Mario, Mercurio, Ciro, Hamel, Ernest, Lavia, Patrizia, Silvestri, Romano
Опубликовано 2014

Toward Highly Potent Cancer Agents by Modulating the C-2 Group of the Arylthioindole Class of Tubulin Polymerization Inhibitors

по La Regina, Giuseppe, Bai, Ruoli, Rensen, Whilelmina Maria, Di Cesare, Erica, Coluccia, Antonio, Piscitelli, Francesco, Famiglini, Valeria, Reggio, Alessia, Nalli, Marianna, Pelliccia, Sveva, Pozzo, Eleonora Da, Costa, Barbara, Granata, Ilaria, Porta, Amalia, Maresca, Bruno, Soriani, Alessandra, Iannitto, Maria Luisa, Santoni, Angela, Li, Junjie, Cona, Marlein Miranda, Chen, Feng, Ni, Yicheng, Brancale, Andrea, Dondio, Giulio, Vultaggio, Stefania, Varasi, Mario, Mercurio, Ciro, Martini, Claudia, Hamel, Ernest, Lavia, Patrizia, Novellino, Ettore, Silvestri, Romano
Опубликовано 2012

New Indole Tubulin Assembly Inhibitors Cause Stable Arrest of Mitotic Progression, Enhanced Stimulation of Natural Killer Cell Cytotoxic Activity, and Repression of Hedgehog-Depend...

по La Regina, Giuseppe, Bai, Ruoli, Coluccia, Antonio, Famiglini, Valeria, Pelliccia, Sveva, Passacantilli, Sara, Mazzoccoli, Carmela, Ruggieri, Vitalba, Verrico, Annalisa, Miele, Andrea, Monti, Ludovica, Nalli, Marianna, Alfonsi, Romina, Di Marcotullio, Lucia, Gulino, Alberto, Ricci, Biancamaria, Soriani, Alessandra, Santoni, Angela, Caraglia, Michele, Porto, Stefania, Pozzo, Eleonora Da, Martini, Claudia, Brancale, Andrea, Marinelli, Luciana, Novellino, Ettore, Vultaggio, Stefania, Varasi, Mario, Mercurio, Ciro, Bigogno, Chiara, Dondio, Giulio, Hamel, Ernest, Lavia, Patrizia, Silvestri, Romano
Опубликовано в: J Med Chem (2015)