Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: A complete structure–activity profile

Por Cacciari, Barbara, Bolcato, Chiara, Spalluto, Giampiero, Klotz, Karl-Norbet, Bacilieri, Magdalena, Deflorian, Francesca, Moro, Stefano
Publicado em 2006

Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: Effect of the N-5 bond type on the affinity and selectivity at the four adenosine receptor subtypes

Por Bolcato, Chiara, Cusan, Claudia, Pastorin, Giorgia, Spalluto, Giampiero, Cacciari, Barbara, Klotz, Karl Norbert, Morizzo, Erika, Moro, Stefano
Publicado em 2007

The Influence of the 1-(3-Trifluoromethyl-Benzyl)-1H-Pyrazole-4-yl Moiety on the Adenosine Receptors Affinity Profile of Pyrazolo[4,3-e][1,2,4]Triazolo[1,5-c]Pyrimidine Derivatives

Por Federico, Stephanie, Redenti, Sara, Sturlese, Mattia, Ciancetta, Antonella, Kachler, Sonja, Klotz, Karl-Norbert, Cacciari, Barbara, Moro, Stefano, Spalluto, Giampiero
Publicado no PLoS One (2015)

Synthesis and pharmacological characterization of a new series of 5,7-disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazine derivatives as adenosine receptor antagonists: A prelimina...

Por Pastorin, Giorgia, Federico, Stephanie, Paoletta, Silvia, Corradino, Marta, Cateni, Francesca, Cacciari, Barbara, Klotz, Karl-Norbert, Gao, Zhan-Guo, Jacobson, Kenneth A., Spalluto, Giampiero, Moro, Stefano
Publicado em 2010

Synthesis and Biological Evaluation of a New Series of 1,2,4-triazolo[1,5-a]-1,3,5-triazines as Human A(2A) Adenosine Receptor Antagonists with Improved Water Solubility

Por Federico, Stephanie, Paoletta, Silvia, Cheong, Siew Lee, Pastorin, Giorgia, Cacciari, Barbara, Stragliotto, Stefano, Klotz, Karl Norbert, Siegel, Jeffrey, Gao, Zhan-Guo, Jacobson, Kenneth A., Moro, Stefano, Spalluto, Giampiero
Publicado em 2011