Drug–Drug Interaction Studies: Regulatory Guidance and An Industry Perspective

द्वारा Prueksaritanont, Thomayant, Chu, Xiaoyan, Gibson, Christopher, Cui, Donghui, Yee, Ka Lai, Ballard, Jeanine, Cabalu, Tamara, Hochman, Jerome
प्रकाशित 2013

Pharmacological validation of a novel nonhuman primate measure of thermal responsivity with utility for predicting analgesic effects

द्वारा Vardigan, Joshua D, Houghton, Andrea K, Lange, Henry S, Adarayan, Emily D, Pall, Parul S, Ballard, Jeanine E, Henze, Darrell A, Uslaner, Jason M
में प्रकाशित J Pain Res (2018)

Application of Pharmacokinetic-Pharmacodynamic Modeling to Inform Translation of In Vitro NaV1.7 Inhibition to In Vivo Pharmacological Response in Non-human Primate

द्वारा Ballard, Jeanine E., Pall, Parul, Vardigan, Joshua, Zhao, Fuqiang, Holahan, Marie A., Kraus, Richard, Li, Yuxing, Henze, Darrell, Houghton, Andrea, Burgey, Christopher S., Gibson, Christopher
में प्रकाशित Pharm Res (2020)

Antagonism of T-type calcium channels inhibits high-fat diet–induced weight gain in mice

द्वारा Uebele, Victor N., Gotter, Anthony L., Nuss, Cindy E., Kraus, Richard L., Doran, Scott M., Garson, Susan L., Reiss, Duane R., Li, Yuxing, Barrow, James C., Reger, Thomas S., Yang, Zhi-Qiang, Ballard, Jeanine E., Tang, Cuyue, Metzger, Joseph M., Wang, Sheng-Ping, Koblan, Kenneth S., Renger, John J.
प्रकाशित 2009

Discovery of Arylsulfonamide Na(v)1.7 Inhibitors: IVIVC, MPO Methods, and Optimization of Selectivity Profile

द्वारा Roecker, Anthony J., Layton, Mark E., Pero, Joseph E., Kelly, Michael J., Greshock, Thomas J., Kraus, Richard L., Li, Yuxing, Klein, Rebecca, Clements, Michelle, Daley, Christopher, Jovanovska, Aneta, Ballard, Jeanine E., Wang, Deping, Zhao, Fuqiang, Brunskill, Andrew P. J., Peng, Xuanjia, Wang, Xiu, Sun, Haiyan, Houghton, Andrea K., Burgey, Christopher S.
में प्रकाशित ACS Med Chem Lett (2021)

Discovery of 4,4-Disubstituted Quinazolin-2-ones as T-Type Calcium Channel Antagonists

द्वारा Barrow, James C., Rittle, Kenneth E., Reger, Thomas S., Yang, Zhi-Qiang, Bondiskey, Phung, McGaughey, Georgia B., Bock, Mark G., Hartman, George D., Tang, Cuyue, Ballard, Jeanine, Kuo, Yuhsin, Prueksaritanont, Thomayant, Nuss, Cindy E., Doran, Scott M., Fox, Steven V., Garson, Susan L., Kraus, Richard L., Li, Yuxing, Marino, Michael J., Kuzmick Graufelds, Valerie, Uebele, Victor N., Renger, John J.
प्रकाशित 2010

Short-Acting T-Type Calcium Channel Antagonists Significantly Modify Sleep Architecture in Rodents

द्वारा Yang, Zhi-Qiang, Schlegel, Kelly-Ann S., Shu, Youheng, Reger, Thomas S., Cube, Rowena, Mattern, Christa, Coleman, Paul J., Small, Jim, Hartman, George D., Ballard, Jeanine, Tang, Cuyue, Kuo, Yuhsin, Prueksaritanont, Thomayant, Nuss, Cindy E., Doran, Scott, Fox, Steve V., Garson, Susan L., Li, Yuxing, Kraus, Richard L., Uebele, Victor N., Taylor, Adekemi B., Zeng, Wei, Fang, Wei, Chavez-Eng, Cynthia, Troyer, Matthew D., Luk, Julie Ann, Laethem, Tine, Cook, William O., Renger, John J., Barrow, James C.
प्रकाशित 2010

Design and Synthesis of Piperazine Sulfonamide Cores Leading to Highly Potent HIV-1 Protease Inhibitors

द्वारा Bungard, Christopher J., Williams, Peter D., Schulz, Jurgen, Wiscount, Catherine M., Holloway, M. Katharine, Loughran, H. Marie, Manikowski, Jesse J., Su, Hua-Poo, Bennett, David J., Chang, Lehua, Chu, Xin-Jie, Crespo, Alejandro, Dwyer, Michael P., Keertikar, Kartik, Morriello, Gregori J., Stamford, Andrew W., Waddell, Sherman T., Zhong, Bin, Hu, Bin, Ji, Tao, Diamond, Tracy L., Bahnck-Teets, Carolyn, Carroll, Steven S., Fay, John F., Min, Xu, Morris, William, Ballard, Jeanine E., Miller, Michael D., McCauley, John A.
में प्रकाशित ACS Med Chem Lett (2017)

Discovery of MK-8718, an HIV Protease Inhibitor Containing a Novel Morpholine Aspartate Binding Group

द्वारा Bungard, Christopher J., Williams, Peter D., Ballard, Jeanine E., Bennett, David J., Beaulieu, Christian, Bahnck-Teets, Carolyn, Carroll, Steve S., Chang, Ronald K., Dubost, David C., Fay, John F., Diamond, Tracy L., Greshock, Thomas J., Hao, Li, Holloway, M. Katharine, Felock, Peter J., Gesell, Jennifer J., Su, Hua-Poo, Manikowski, Jesse J., McKay, Daniel J., Miller, Mike, Min, Xu, Molinaro, Carmela, Moradei, Oscar M., Nantermet, Philippe G., Nadeau, Christian, Sanchez, Rosa I., Satyanarayana, Tummanapalli, Shipe, William D., Singh, Sanjay K., Truong, Vouy Linh, Vijayasaradhi, Sivalenka, Wiscount, Catherine M., Vacca, Joseph P., Crane, Sheldon N., McCauley, John A.
में प्रकाशित ACS Med Chem Lett (2016)