Fragment-Based Optimization of Small Molecule CXCL12 Inhibitors for Antagonizing the CXCL12/CXCR4 Interaction

Por Ziarek, Joshua J., Liu, Yan, Smith, Emmanuel, Zhang, Guolin, Peterson, Francis C., Chen, Jun, Yu, Yongping, Chen, Yu, Volkman, Brian F., Li, Rongshi
Publicado em 2012

Insights into the structure-activity relationship of the anticancer compound ZJ-101, a derivative of marine natural product superstolide A: a role played by the lactone moiety

Por Qiu, Haibo, Qian, Shan, Head, Sarah A., Liu, Jun O., Jin, Zhendong
Publicado no Bioorg Med Chem Lett (2016)

Advances in the discovery of cathepsin K inhibitors on bone resorption

Por Lu, Jun, Wang, Maolin, Wang, Ziyue, Fu, Zhongqi, Lu, Aiping, Zhang, Ge
Publicado no J Enzyme Inhib Med Chem (2018)

Green synthesis of a typical chiral stationary phase of cellulose-tris(3, 5-dimethylphenylcarbamate)

Por Liu, Run-Qiang, Bai, Lian-yang, Zhang, Yi-Jun, Zhang, Yu-Ping
Publicado em 2013

The dependence of Ni-Fe bioxide composites nanoparticles on the FeCl(2) solution used

Por Lin, Yueqiang, Li, Jian, Lin, Lihua, Liu, Xiaodong, Chen, Longlong, Fu, Jun
Publicado em 2012

Synthesis and biological evaluation of 1, 3-dihydroxyxanthone mannich base derivatives as anticholinesterase agents

Por Qin, Jiangke, Lan, Wenli, Liu, Zhong, Huang, Jun, Tang, Huang, Wang, Hengshan
Publicado em 2013

Structure Guided Development of Novel Thymidine Mimetics targeting Pseudomonas aeruginosa Thymidylate Kinase: from Hit to Lead Generation

Por Choi, Jun Yong, Plummer, Mark S., Starr, Jeremy, Desbonnet, Charlene R., Soutter, Holly, Chang, Jeanne, Miller, J. Richard, Dillman, Keith, Miller, Alita A., Roush, William R.
Publicado em 2012

Development of a dual-wavelength fluorescent nanoprobe for in vivo and in vitro cell tracking consecutively

Por Vu, Hong, Zhou, Jun, Huang, Yihui, Hakamivala, Amirhossein, Khang, Min Kyung, Tang, Liping
Publicado no Bioorg Med Chem (2019)

Regiospecific and conformationally restrained analogs of melphalan and DL-2-NAM-7 and their affinities for the large neutral amino acid transporter (system LAT1) of the blood–brain...

Por Matharu, Jyothi, Oki, Jun, Worthen, David R., Smith, Quentin R., Crooks, Peter A.
Publicado em 2010

SAR by Inter-Ligand nuclear Overhauser Effects (ILOEs) based discovery of acylsulfonamide compounds active against Bcl-x(L) and Mcl-1

Por Rega, Michele F., Wu, Bainan, Wei, Jun, Zhang, Ziming, Cellitti, Jason F., Pellecchia, Maurizio
Publicado em 2011

Three novel oligosaccharides synthesized using Thermoanaerobacter brockii kojibiose phosphorylase

Por Takahashi, Natsuko, Fukushi, Eri, Onodera, Shuichi, Benkeblia, Noureddine, Nishimoto, Tomoyuki, Kawabata, Jun, Shiomi, Norio
Publicado em 2007

Structural analysis of three novel trisaccharides isolated from the fermented beverage of plant extracts

Por Okada, Hideki, Fukushi, Eri, Yamamori, Akira, Kawazoe, Naoki, Onodera, Shuichi, Kawabata, Jun, Shiomi, Norio
Publicado em 2009

Quantitative analysis of the major constituents in Chinese medicinal preparation SuoQuan formulae by ultra fast high performance liquid chromatography/quadrupole tandem mass spectr...

Por Chen, Feng, Li, Hai-long, Li, Yong-Hui, Tan, Yin-Feng, Zhang, Jun-Qing
Publicado em 2013

Synthesis and biological evaluation of novel 7-hydroxy-4-phenylchromen-2-one–linked to triazole moieties as potent cytotoxic agents

Por Liu, Chuan-Feng, Shen, Qing-Kun, Li, Jia-Jun, Tian, Yu-Shun, Quan, Zheshan
Publicado no J Enzyme Inhib Med Chem (2017)

Redox Potentials, Laccase Oxidation, and Antilarval Activities of Substituted Phenols

Por Prasain, Keshar, Nguyen, Thi D. T., Gorman, Maureen J., Barrigan, Lydia M., Peng, Zeyu, Kanost, Michael R., Syed, Lateef U., Li, Jun, Zhu, Kun Yan, Hua, Duy H.
Publicado em 2012

Identificaiton of Shc Src Homology 2 Domain-Binding Peptoid – Peptide Hybrids

Por Choi, Won Jun, Kim, Sung Eun, Stephen, Andrew G., Weidlich, Iwona, Giubellino, Alessio, Liu, Fa, Worthy, Karen M., Bindu, Lakshman, Fivash, Matthew J., Nicklaus, Marc C., Bottaro, Donald P., Fisher, Robert J., Burke, Terrence R.
Publicado em 2009

Discovery of Phenylaminopyridine Derivatives as Novel HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors

Por Kim, Junwon, Lee, Doohyun, Park, Changmin, So, Wonyoung, Jo, Mina, Ok, Taedong, Kwon, Jeongjin, Kong, Sunju, Jo, Suyeon, Kim, Youngmi, Choi, Jihyun, Kim, Hyoung Cheul, Ko, Yoonae, Choi, Inhee, Park, Youngsam, Yoon, Jaewan, Ju, Moon Kyeong, Kim, Junghwan, Han, Sung-Jun, Kim, Tae-Hee, Cechetto, Jonathan, Nam, Jiyoun, Sommer, Peter, Liuzzi, Michel, Lee, Jinhwa, No, Zaesung
Publicado em 2012

Rational design of potent and selective inhibitors of an epoxide hydrolase virulence factor from Pseudomonas aeruginosa

Por Kitamura, Seiya, Hvorecny, Kelli L., Niu, Jun, Hammock, Bruce D., Madden, Dean R., Morisseau, Christophe
Publicado no J Med Chem (2016)

Efficient synthesis and biological evaluation of epiceanothic acid and related compounds

Por Zhang, Pu, Xu, Li, Qian, Keduo, Liu, Jun, Zhang, Luyong, Lee, Kuo-Hsiung, Sun, Hongbin
Publicado em 2010

Itraconazole Side Chain Analogues: Structure–Activity Relationship Studies for Inhibition of Endothelial Cell Proliferation, Vascular Endothelial Growth Factor Receptor 2 (VEGFR2)...

Por Shi, Wei, Nacev, Benjamin A., Aftab, Blake T., Head, Sarah, Rudin, Charles M., Liu, Jun O.
Publicado em 2011