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Hexose-6-phosphate dehydrogenase blockade reverses prostate cancer drug resistance in xenograft models by glucocorticoid inactivation

Prostate cancer resistance to next-generation hormonal treatment with enzalutamide is a major problem and eventuates into disease lethality. Biologically active glucocorticoids that stimulate glucocorticoid receptor (GR) have an 11β-OH moiety and resistant tumors exhibit loss of 11β-HSD2, the oxidat...

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Dettagli Bibliografici
Pubblicato in:Sci Transl Med
Autori principali: Jianneng Li, Berk, Michael, Alyamani, Mohammad, Sabharwal, Navin, Goins, Christopher, Alvarado, Joseph, Baratchian, Mehdi, Zhu, Ziqi, Stauffer, Shaun, Klein, Eric A., Sharifi, Nima
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC8319670/
https://ncbi.nlm.nih.gov/pubmed/34039740
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/scitranslmed.abe8226
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