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Differential Inhibition of Equilibrative Nucleoside Transporter 1 (ENT1) Activity by Tyrosine Kinase Inhibitors

BACKGROUND AND OBJECTIVES: Equilibrative nucleoside transporter (ENT) 1 is a widely-expressed drug transporter, handling nucleoside analogues as well as endogenous nucleosides. ENT1 has been postulated to be inhibited by some marketed tyrosine kinase inhibitors (TKIs). To obtain insights into this p...

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Detalles Bibliográficos
Publicado en:Eur J Drug Metab Pharmacokinet
Main Authors: Jouan, Elodie, Moreau, Amélie, Bruyere, Arnaud, Alim, Karima, Denizot, Claire, Parmentier, Yannick, Fardel, Olivier
Formato: Artigo
Idioma:Inglês
Publicado: Springer International Publishing 2021
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC8286641/
https://ncbi.nlm.nih.gov/pubmed/34275128
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s13318-021-00703-2
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