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Subtype-selective mechanisms of negative allosteric modulators binding to group I metabotropic glutamate receptors

Group I metabotropic glutamate receptors (mGlu(1) and mGlu(5)) are promising targets for multiple psychiatric and neurodegenerative disorders. Understanding the subtype selectivity of mGlu(1) and mGlu(5) allosteric sites is essential for the rational design of novel modulators with single- or dual-t...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Acta Pharmacol Sin
Egile Nagusiak: Fu, Ting-ting, Tu, Gao, Ping, Meng, Zheng, Guo-xun, Yang, Feng-yuan, Yang, Jing-yi, Zhang, Yang, Yao, Xiao-jun, Xue, Wei-wei, Zhu, Feng
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Springer Singapore 2020
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC8285414/
https://ncbi.nlm.nih.gov/pubmed/33122823
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41401-020-00541-z
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