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Cyclopropyl-containing positive allosteric modulators of metabotropic glutamate receptor subtype 5

Positive allosteric modulators (PAM) binding to the transmembrane (TM) domain of metabotropic glutamate receptor 5 (mGluR5) are promising therapeutic agents for psychiatric disorders and traumatic brain injury (TBI). Novel PAMs based on a trans-2-phenylcyclopropane amide scaffold have been designed...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Lakkaraju, Sirish K., Mbatia, Hannah, Hanscom, Marie, Zhao, Zaorui, Wu, Junfang, Stoica, Bogdan, MacKerell, Alexander D., Faden, Alan I., Xue, Fengtian
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4690453/
https://ncbi.nlm.nih.gov/pubmed/25937015
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.04.042
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