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Synthesis and Biological Activity of Conformationally Restricted Indole-based Inhibitors of Neurotropic Alphavirus Replication: Generation of a Three-Dimensional Pharmacophore

We have previously reported the development of indole-based CNS-active antivirals for the treatment of neurotropic alphavirus infection, but further optimization is impeded by a lack of knowledge of the molecular target and binding site. Herein we describe the design, synthesis, and evaluation of a...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Barraza, Scott J., Sindac, Janice A., Dobry, Craig J., Delekta, Philip C., Lee, Pil H., Miller, David J., Larsen, Scott D.
Formato: Artigo
Idioma:Inglês
Publicado em: 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8272561/
https://ncbi.nlm.nih.gov/pubmed/34098081
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2021.128171
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