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High-Throughput Quality Control Assay for the Solid-Phase Synthesis of DNA-Encoded Libraries of Macrocycles

There is considerable interest in the development of libraries of scaffold-diverse macrocycles as a source of ligands for difficult targets, such as protein–protein interaction surfaces. A classic problem in the synthesis of high-quality macrocyclic libraries is that some linear precursors will cycl...

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Publicat a:Angew Chem Int Ed Engl
Autors principals: Roy, Animesh, Koesema, Eric, Kodadek, Thomas
Format: Artigo
Idioma:Inglês
Publicat: 2021
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8193836/
https://ncbi.nlm.nih.gov/pubmed/33682283
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.202100230
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