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Computational strategy for intrinsically disordered protein ligand design leads to the discovery of p53 transactivation domain I binding compounds that activate the p53 pathway

Intrinsically disordered proteins or intrinsically disordered regions (IDPs) have gained much attention in recent years due to their vital roles in biology and prevalence in various human diseases. Although IDPs are perceived as attractive therapeutic targets, rational drug design targeting IDPs rem...

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Dettagli Bibliografici
Pubblicato in:Chem Sci
Autori principali: Ruan, Hao, Yu, Chen, Niu, Xiaogang, Zhang, Weilin, Liu, Hanzhong, Chen, Limin, Xiong, Ruoyao, Sun, Qi, Jin, Changwen, Liu, Ying, Lai, Luhua
Natura: Artigo
Lingua:Inglês
Pubblicazione: The Royal Society of Chemistry 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC8179352/
https://ncbi.nlm.nih.gov/pubmed/34164069
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0sc04670a
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