Chargement en cours...

One-pot thiol–amine bioconjugation to maleimides: simultaneous stabilisation and dual functionalisation

Maleimide chemistry is widely used in the site-selective modification of proteins. However, hydrolysis of the resultant thiosuccinimides is required to provide robust stability to the bioconjugates. Herein, we present an alternative approach that affords simultaneous stabilisation and dual functiona...

Description complète

Enregistré dans:
Détails bibliographiques
Publié dans:Chem Sci
Auteurs principaux: Wall, Archie, Wills, Alfie G., Forte, Nafsika, Bahou, Calise, Bonin, Lisa, Nicholls, Karl, Ma, Michelle T., Chudasama, Vijay, Baker, James R.
Format: Artigo
Langue:Inglês
Publié: The Royal Society of Chemistry 2020
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC8162801/
https://ncbi.nlm.nih.gov/pubmed/34094388
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0sc05128d
Tags: Ajouter un tag
Pas de tags, Soyez le premier à ajouter un tag!