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Coordinating bioorthogonal reactions with two tumor-microenvironment-responsive nanovehicles for spatiotemporally controlled prodrug activation

Precise activation of prodrugs in tumor tissues is critical to ensuring specific antitumor efficacy, meanwhile reducing the serious adverse effects. Here, a spatiotemporally controlled prodrug activation strategy was provided by integrating the inverse electron demand Diels–Alder (IEDDA) reaction wi...

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Publicado en:Chem Sci
Main Authors: Zuo, Liping, Ding, Jingjing, Li, Changkun, Lin, Feng, Chen, Peng R., Wang, Peilin, Lu, Guihong, Zhang, Jinfeng, Huang, Li-Li, Xie, Hai-Yan
Formato: Artigo
Idioma:Inglês
Publicado: The Royal Society of Chemistry 2020
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC8150104/
https://ncbi.nlm.nih.gov/pubmed/34123305
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c9sc05036a
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