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Exploring naltrexamine derivatives featuring azaindole moiety via nitrogen-walk approach to investigate their in vitro pharmacological profiles at the mu opioid receptor

In the present work, we reported the application of a nitrogen-walk approach on developing a series of novel opioid ligands containing an azaindole moiety at the C6-position of the epoxymorphinan skeleton. In vitro study results showed that introducing a nitrogen atom around the indole moiety not on...

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Publicat a:Bioorg Med Chem Lett
Autors principals: Ma, Hongguang, Wang, Huiqun, Gillespie, James C., Mendez, Rolando E., Selley, Dana E., Zhang, Yan
Format: Artigo
Idioma:Inglês
Publicat: 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8113153/
https://ncbi.nlm.nih.gov/pubmed/33766769
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2021.127953
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