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Mixed Kappa/Mu Opioid Receptor Agonists: The 6β-Naltrexamines
Ligands from the naltrexamine series have consistently demonstrated agonist activity at kappa opioid receptors (KOR), with varying activity at the mu opioid receptor (MOR). Various 6β-cinnamoylamino derivatives were made with the aim of generating ligands with a KOR agonist/MOR partial agonist profi...
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| Главные авторы: | , , , , , , , , |
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| Формат: | Artigo |
| Язык: | Inglês |
| Опубликовано: |
2009
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| Предметы: | |
| Online-ссылка: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3070388/ https://ncbi.nlm.nih.gov/pubmed/19253970 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm8015552 |
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