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Targeting Bromodomain and Extraterminal Proteins for Drug Discovery: From Current Progress to Technological Development

Bromodomain and extraterminal (BET) proteins bind acetylated lysine residues in histones and nonhistone proteins via tandem bromodomains and regulate chromatin dynamics, cellular processes, and disease procession. Thus targeting BET proteins is a promising strategy for treating various diseases, esp...

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Bibliographic Details
Published in:J Med Chem
Main Authors: Tang, Pan, Zhang, Jifa, Liu, Jie, Chiang, Cheng-Ming, Ouyang, Liang
Format: Artigo
Language:Inglês
Published: 2021
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC8106541/
https://ncbi.nlm.nih.gov/pubmed/33616410
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.0c01487
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