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Targeting Bromodomain and Extraterminal Proteins for Drug Discovery: From Current Progress to Technological Development

Bromodomain and extraterminal (BET) proteins bind acetylated lysine residues in histones and nonhistone proteins via tandem bromodomains and regulate chromatin dynamics, cellular processes, and disease procession. Thus targeting BET proteins is a promising strategy for treating various diseases, esp...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:J Med Chem
Hauptverfasser: Tang, Pan, Zhang, Jifa, Liu, Jie, Chiang, Cheng-Ming, Ouyang, Liang
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2021
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC8106541/
https://ncbi.nlm.nih.gov/pubmed/33616410
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.0c01487
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