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Effect of four ABCB1 genetic polymorphisms on the accumulation of darunavir in HEK293 recombinant cell lines

The intracellular penetration of darunavir, a second-generation HIV protease inhibitor, is limited by the activity of the efflux P-glycoprotein (ABCB1). ABCB1 expression and/or activity levels can vary between individuals due to genetic polymorphisms including the c.1199G>A, c.1236C>T, c.2677G...

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Detaylı Bibliyografya
Yayımlandı:Sci Rep
Asıl Yazarlar: Stillemans, Gabriel, Djokoto, Happy Phanio, Delongie, Kévin-Alexandre, El-Hamdaoui, Halima, Panin, Nadtha, Haufroid, Vincent, Elens, Laure
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Nature Publishing Group UK 2021
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC8076219/
https://ncbi.nlm.nih.gov/pubmed/33903659
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-021-88365-7
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