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Evaluation of Hsp90 and mTOR inhibitors as potential drugs for the treatment of TSC1/TSC2 deficient cancer

Inactivating mutations in either TSC1 or TSC2 cause Tuberous Sclerosis Complex, an autosomal dominant disorder, characterized by multi-system tumor and hamartoma development. Mutation and loss of function of TSC1 and/or TSC2 also occur in a variety of sporadic cancers, and rapamycin and related drug...

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Библиографические подробности
Опубликовано в: :PLoS One
Главные авторы: Mrozek, Evelyn M., Bajaj, Vineeta, Guo, Yanan, Malinowska, Izabela A., Zhang, Jianming, Kwiatkowski, David J.
Формат: Artigo
Язык:Inglês
Опубликовано: Public Library of Science 2021
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC8064564/
https://ncbi.nlm.nih.gov/pubmed/33891611
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0248380
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