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The Inclusion of Tolfenamic Acid into Cyclodextrins Stimulated by Microenvironmental pH Modification as a Way to Increase the Anti-Migraine Effect
PURPOSE: The poorly soluble nonsteroidal anti-inflammatory drug (NSAID), tolfenamic acid (TA), was studied to maximize its solubility, permeability through biological membranes, and pharmacological activity. METHODS: A mixture with magnesium stearate (MS) – microenvironment pH-modifier was prepared,...
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| Опубликовано в: : | J Pain Res |
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| Главные авторы: | , , , , , , , , , |
| Формат: | Artigo |
| Язык: | Inglês |
| Опубликовано: |
Dove
2021
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| Предметы: | |
| Online-ссылка: | https://ncbi.nlm.nih.gov/pmc/articles/PMC8055370/ https://ncbi.nlm.nih.gov/pubmed/33883930 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2147/JPR.S295795 |
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