Discovery of a Remarkable Methyl Shift Effect in the Vanilloid Activity of Triterpene Amides

[Image: see text] As part of a study on triterpenoid conjugates, the dietary pentacyclic triterpenoids oleanolic (2a) and ursolic acids (3a) were coupled with vanillamine, and the resulting amides (2b and 3b, respectively) were assayed for activity on the vanilloid receptor TRPV1. Despite a structur...

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Bibliografische gegevens
Gepubliceerd in:J Nat Prod
Hoofdauteurs: Vitale, Rosa Maria, Avonto, Cristina, Del Prete, Danilo, Moriello, Aniello Schiano, Amodeo, Pietro, Appendino, Giovanni, De Petrocellis, Luciano
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: American Chemical Society and American Society of Pharmacognosy 2020
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC8016363/
https://ncbi.nlm.nih.gov/pubmed/33136399
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jnatprod.0c00639
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