Effective microwave-assisted approach to 1,2,3-triazolobenzodiazepinones via tandem Ugi reaction/catalyst-free intramolecular azide–alkyne cycloaddition

A novel catalyst-free synthetic approach to 1,2,3-triazolobenzodiazepinones has been developed and optimized. The Ugi reaction of 2-azidobenzaldehyde, various amines, isocyanides, and acids followed by microwave-assisted intramolecular azide–alkyne cycloaddition (IAAC) gave a series of target hetero...

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Detalhes bibliográficos
Publicado no:Beilstein J Org Chem
Main Authors: Mazur, Maryna O, Zhelavskyi, Oleksii S, Zviagin, Eugene M, Shishkina, Svitlana V, Musatov, Vladimir I, Kolosov, Maksim A, Shvets, Elena H, Andryushchenko, Anna Yu, Chebanov, Valentyn A
Formato: Artigo
Idioma:Inglês
Publicado em: Beilstein-Institut 2021
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Full Research Paper
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7961865/
https://ncbi.nlm.nih.gov/pubmed/33777243
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.17.57
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