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A Diverse Range of Hemozoin Inhibiting Scaffolds Act on Plasmodium falciparum as Heme Complexes
A diverse series of hemozoin-inhibiting quinolines, benzamides, triarylimidazoles, quinazolines, benzimidazoles, benzoxazoles and benzothiazoles have been found to lead to exchangeable heme in cultured Plasmodium falciparum (NF54) that ranged over an order of magnitude at the IC(50). Surprisingly, l...
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| Publicat a: | ACS Infect Dis |
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| Autors principals: | , , , , , , |
| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
2021
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7948512/ https://ncbi.nlm.nih.gov/pubmed/33430579 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.0c00680 |
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