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Structural basis of antagonizing the vitamin K catalytic cycle for anticoagulation

Vitamin K antagonists are widely used anticoagulants targeting vitamin K epoxide reductases (VKOR), a unique family of integral membrane enzymes. To elucidate their catalytic cycle and inhibitory mechanism, here we report eleven x-ray crystal structures of human VKOR and a VKOR-like paralog with sub...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Science
Egile Nagusiak: Liu, Shixuan, Li, Shuang, Shen, Guomin, Sukumar, Narayanasami, Krezel, Andrzej M., Li, Weikai
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2020
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC7946407/
https://ncbi.nlm.nih.gov/pubmed/33154105
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/science.abc5667
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