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Methods for the discovery of small molecules to monitor and perturb the activity of the human proteasome

Regulating protein production and degradation is critical to maintaining cellular homeostasis. The proteasome is a key player in keeping proteins at the proper levels. However, proteasome activity can be altered in certain disease states, such as blood cancers and neurodegenerative diseases. Cancers...

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Библиографические подробности
Опубликовано в: :Future Med Chem
Главные авторы: Maresh, Marianne E, Salazar-Chaparro, Andres F, Trader, Darci J
Формат: Artigo
Язык:Inglês
Опубликовано: Newlands Press Ltd 2020
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC7857359/
https://ncbi.nlm.nih.gov/pubmed/33275045
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4155/fmc-2020-0288
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