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Intrabacterial Metabolism Obscures the Successful Prediction of an InhA Inhibitor of Mycobacterium tuberculosis

Tuberculosis, caused by Mycobacterium tuberculosis (M. tuberculosis), kills 1.6 million people annually. To bridge the gap between structure- and cell-based drug discovery strategies, we are pioneering a computer-aided discovery paradigm that merges structure-based virtual screening with ligand-base...

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Podrobná bibliografie
Vydáno v:ACS Infect Dis
Hlavní autoři: Wang, Xin, Perryman, Alexander L., Li, Shao-Gang, Paget, Steve D., Stratton, Thomas P., Lemenze, Alex, Olson, Arthur J., Ekins, Sean, Kumar, Pradeep, Freundlich, Joel S.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2019
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7801736/
https://ncbi.nlm.nih.gov/pubmed/31625383
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.9b00295
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