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Intrabacterial Metabolism Obscures the Successful Prediction of an InhA Inhibitor of Mycobacterium tuberculosis

Tuberculosis, caused by Mycobacterium tuberculosis (M. tuberculosis), kills 1.6 million people annually. To bridge the gap between structure- and cell-based drug discovery strategies, we are pioneering a computer-aided discovery paradigm that merges structure-based virtual screening with ligand-base...

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Detalles Bibliográficos
Publicado en:ACS Infect Dis
Main Authors: Wang, Xin, Perryman, Alexander L., Li, Shao-Gang, Paget, Steve D., Stratton, Thomas P., Lemenze, Alex, Olson, Arthur J., Ekins, Sean, Kumar, Pradeep, Freundlich, Joel S.
Formato: Artigo
Idioma:Inglês
Publicado: 2019
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7801736/
https://ncbi.nlm.nih.gov/pubmed/31625383
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.9b00295
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