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Inhibiting Sialidase-Induced TGF-β1 Activation Attenuates Pulmonary Fibrosis in Mice

The active form of transforming growth factor-β1 (TGF-β1) plays a key role in potentiating fibrosis. TGF-β1 is sequestered in an inactive state by a latency-associated glycopeptide (LAP). Sialidases (also called neuraminidases (NEU)) cleave terminal sialic acids from glycoconjugates. The sialidase N...

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Publicado en:J Pharmacol Exp Ther
Autores principales: Karhadkar, Tejas R., Meek, Thomas D., Gomer, Richard H.
Formato: Artigo
Lenguaje:Inglês
Publicado: The American Society for Pharmacology and Experimental Therapeutics 2021
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7788355/
https://ncbi.nlm.nih.gov/pubmed/33144389
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.120.000258
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