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Ligand-Dependent Effects of Methionine-8 Oxidation in Parathyroid Hormone Peptide Analogues

LA-PTH is a long-acting parathyroid hormone (PTH) peptide analogue in preclinical development for hypoparathyroidism (HP). Like native PTH, LA-PTH contains a methionine at position 8 (Met8) that is predicted to be critical for function. We assessed the impact of Met oxidation on the functional prope...

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Bibliografski detalji
Izdano u:Endocrinology
Glavni autori: Daley, Eileen J, Khatri, Ashok, Dean, Thomas, Vilardaga, Jean-Pierre, Zaidi, Saheem A, Katritch, Vsevolod, Gardella, Thomas J
Format: Artigo
Jezik:Inglês
Izdano: Oxford University Press 2020
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Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7774776/
https://ncbi.nlm.nih.gov/pubmed/33242090
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1210/endocr/bqaa216
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