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Molecular Docking Simulations on Histone Deacetylases (HDAC)-1 and -2 to Investigate the Flavone Binding

Histone modifications through acetylation are fundamental for remodelling chromatin and consequently activating gene expression. The imbalance between acetylation and deacetylation activity causes transcriptional dysregulation associated with several disorders. Flavones, small molecules of plant ori...

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Dettagli Bibliografici
Pubblicato in:Biomedicines
Autori principali: Scafuri, Bernardina, Bontempo, Paola, Altucci, Lucia, De Masi, Luigi, Facchiano, Angelo
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7761979/
https://ncbi.nlm.nih.gov/pubmed/33291755
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biomedicines8120568
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