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Discovery of Potent Indenoisoquinoline Topoisomerase I Poisons Lacking the 3-Nitro Toxicophore

3-Nitroindenoisoquinoline human topoisomerase IB (Top1) poisons have potent antiproliferative effects on cancer cells. The undesirable nitro toxicophore could hypothetically be replaced by other functional groups that would retain the desired biological activities and minimize potential safety risks...

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Détails bibliographiques
Publié dans:J Med Chem
Auteurs principaux: Beck, Daniel E., Abdelmalak, Monica, Lv, Wei, Reddy, P. V. Narasimha, Tender, Gabrielle S., O’Neill, Elizaveta, Agama, Keli, Marchand, Christophe, Pommier, Yves, Cushman, Mark
Format: Artigo
Langue:Inglês
Publié: 2015
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7753975/
https://ncbi.nlm.nih.gov/pubmed/25909279
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b00303
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