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Interfacial inhibitors

Targeting macromolecular interface is a general mechanism by which natural products inactivate macromolecular complexes by stabilizing normally transient intermediates. Demonstrating interfacial inhibition mechanism ultimately relies on the resolution of drug-macromolecule structures. This review fo...

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Detalles Bibliográficos
Publicado en:Bioorg Med Chem Lett
Main Authors: Pommier, Yves, Kiselev, Evgeny, Marchand, Christophe
Formato: Artigo
Idioma:Inglês
Publicado: 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7747010/
https://ncbi.nlm.nih.gov/pubmed/26235949
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.07.032
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