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Thioamide Substitution Selectively Modulates Proteolysis and Receptor Activity of Therapeutic Peptide Hormones

Peptide hormones are attractive as injectable therapeutics and imaging agents, but they often require extensive modification by mutagenesis and/or chemical synthesis to prevent rapid in vivo degradation. Alternatively, the single atom, O-to-S modification of peptide backbone thioamidation has the po...

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Bibliografske podrobnosti
izdano v:J Am Chem Soc
Main Authors: Chen, Xing, Mietlicki-Baase, Elizabeth G., Barrett, Taylor M., McGrath, Lauren E., Koch-Laskowski, Kieran, Ferrie, John J., Hayes, Matthew R., Petersson, E. James
Format: Artigo
Jezik:Inglês
Izdano: 2017
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC7744120/
https://ncbi.nlm.nih.gov/pubmed/29130686
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.7b08417
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