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Structural properties and anticoagulant/cytotoxic activities of heterochiral enantiomeric thrombin binding aptamer (TBA) derivatives

The thrombin binding aptamer (TBA) possesses promising antiproliferative properties. However, its development as an anticancer agent is drastically impaired by its concomitant anticoagulant activity. Therefore, suitable chemical modifications in the TBA sequence would be required in order to preserv...

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Publicat a:Nucleic Acids Res
Autors principals: Virgilio, Antonella, Esposito, Veronica, Pecoraro, Annalisa, Russo, Annapina, Vellecco, Valentina, Pepe, Antonietta, Bucci, Mariarosaria, Russo, Giulia, Galeone, Aldo
Format: Artigo
Idioma:Inglês
Publicat: Oxford University Press 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7736819/
https://ncbi.nlm.nih.gov/pubmed/33270863
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/nar/gkaa1109
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