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An Optimal “Click” Formulation Strategy for Antibody-Drug Conjugate Synthesis

As a versatile reaction for bioconjugation, Cu(I)-catalyzed alkyne-azide cycloaddition (CuAAC) has enormous potential in the synthesis of antibody-drug conjugates (ADCs). In order to optimize CuAAC-based ADC synthesis, we characterized kinetically different formulation processes by mimicking ADC syn...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem
Main Authors: Vatansever, Erol C., Kang, Jeffrey, Tuley, Alfred, Ward, E. Sally, Liu, Wenshe Ray
Formato: Artigo
Idioma:Inglês
Publicado em: 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7736079/
https://ncbi.nlm.nih.gov/pubmed/33071032
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2020.115808
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