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5′-O-Aliphatic and amino acid ester prodrugs of (−)-β-d-(2R,4R)-dioxolane-thymine (DOT): Synthesis, anti-HIV activity, cytotoxicity and stability studies

A series of (−)-β-d-(2R,4R)-dioxolane-thymine-5′-O-aliphatic acid esters as well as amino acid esters were synthesized as prodrugs of (−)-β-d-(2R,4R)-dioxolane-thymine (DOT). The compounds were evaluated for anti-HIV activity against HIV-1(LAI) in human peripheral blood mononuclear (PBM) cells as we...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem
Main Authors: Liang, Yuzeng, Sharon, Ashoke, Grier, Jason P., Rapp, Kimberly L., Schinazi, Raymond F., Chu, Chung K.
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7734618/
https://ncbi.nlm.nih.gov/pubmed/19153047
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2008.10.078
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