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Identifying OXA-48 Carbapenemase Inhibitors Using DNA-Encoded Chemical Libraries

Bacterial resistance to β-lactam antibiotics is largely mediated by β-lactamases, which catalyze the hydrolysis of these drugs and continue to emerge in response to antibiotic use. β-lactamases that hydrolyze the last resort carbapenem class of β-lactam antibiotics (carbapenemases) are a growing glo...

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Detalhes bibliográficos
Publicado no:ACS Infect Dis
Main Authors: Taylor, Doris Mia, Anglin, Justin, Park, Suhyeorn, Ucisik, Melek N., Faver, John C., Simmons, Nicholas, Jin, Zhuang, Palaniappan, Murugesan, Nyshadham, Pranavanand, Li, Feng, Campbell, James, Hu, Liya, Sankaran, Banumathi, Prasad, B.V. Venkataram, Huang, Hongbing, Matzuk, Martin M., Palzkill, Timothy
Formato: Artigo
Idioma:Inglês
Publicado em: 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7673237/
https://ncbi.nlm.nih.gov/pubmed/32182432
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.0c00015
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