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Peptidic boronic acid Plasmodium falciparum SUB1 inhibitors with improved selectivity over human proteasome

Plasmodium falciparum subtilisin-like serine protease 1 (PfSUB1) is essential for egress of invasive merozoite forms of the parasite, rendering PfSUB1 an attractive antimalarial target. Here we report studies aimed to improve drug-like properties of peptidic boronic acid PfSUB1 inhibitors including...

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Publicado en:J Med Chem
Autores principales: Withers-Martinez, Chrislaine, Lidumniece, Elina, Hackett, Fiona, Collins, Christine R., Taha, Zahie, Blackman, Michael J., Jirgensons, Aigars
Formato: Artigo
Lenguaje:Inglês
Publicado: 2024
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7616463/
https://ncbi.nlm.nih.gov/pubmed/39051854
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.4c01005
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