Carregant...

Peptidic boronic acid Plasmodium falciparum SUB1 inhibitors with improved selectivity over human proteasome

Plasmodium falciparum subtilisin-like serine protease 1 (PfSUB1) is essential for egress of invasive merozoite forms of the parasite, rendering PfSUB1 an attractive antimalarial target. Here we report studies aimed to improve drug-like properties of peptidic boronic acid PfSUB1 inhibitors including...

Descripció completa

Guardat en:
Dades bibliogràfiques
Publicat a:J Med Chem
Autors principals: Withers-Martinez, Chrislaine, Lidumniece, Elina, Hackett, Fiona, Collins, Christine R., Taha, Zahie, Blackman, Michael J., Jirgensons, Aigars
Format: Artigo
Idioma:Inglês
Publicat: 2024
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7616463/
https://ncbi.nlm.nih.gov/pubmed/39051854
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.4c01005
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!