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Making the switch: The role of Gq in driving GRK selectivity at GPCRs

Selective engagement of signal transducers such as G proteins and β-arrestins with GPCRs upon stimulation with biased agonists is thought to be due to distinct receptor conformations. Kawakami et al. propose an additional mechanism whereby activation of Gq determines GPCR kinase subtype selectivity...

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Bibliographic Details
Published in:Sci Signal
Main Authors: Sarma, Parishmita, Saha, Shirsha, Shukla, Arun K.
Format: Artigo
Language:Inglês
Published: 2022
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC7612787/
https://ncbi.nlm.nih.gov/pubmed/35316098
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/scisignal.abo4949
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