Llwytho...

Development and biological investigations of hypoxia-sensitive prodrugs of the tyrosine kinase inhibitor crizotinib

Despite the huge success of tyrosine kinase inhibitors as anticancer agents, severe side effects are a major problem. In order to overcome this drawback, the first hypoxia-activatable 2-nitroimidazole-based prodrugs of the clinically approved ALK and c-MET inhibitor crizotinib were developed. The 2-...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:Bioorg Chem
Prif Awduron: Bielec, Bjoern, Schueffl, Hemma, Terenzi, Alessio, Berger, Walter, Heffeter, Petra, Keppler, Bernhard K., Kowol, Christian R.
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2020
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC7611434/
https://ncbi.nlm.nih.gov/pubmed/32229347
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bioorg.2020.103778
Tagiau: Ychwanegu Tag
Dim Tagiau, Byddwch y cyntaf i dagio'r cofnod hwn!