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Repurposing Heparin as Antimalarial: Evaluation of Multiple Modifications Toward In Vivo Application

Heparin is a promising antimalarial drug due to its activity in inhibiting Plasmodium invasion of red blood cells and to the lack of resistance evolution by the parasite against it, but its potent anticoagulant activity is preventing the advance of heparin along the clinical pipeline. We have determ...

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Publicat a:Pharmaceutics
Autors principals: Lantero, Elena, Aláez-Versón, Carlos Raúl, Romero, Pilar, Sierra, Teresa, Fernàndez-Busquets, Xavier
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7557421/
https://ncbi.nlm.nih.gov/pubmed/32872434
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics12090825
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