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Repurposing Heparin as Antimalarial: Evaluation of Multiple Modifications Toward In Vivo Application

Heparin is a promising antimalarial drug due to its activity in inhibiting Plasmodium invasion of red blood cells and to the lack of resistance evolution by the parasite against it, but its potent anticoagulant activity is preventing the advance of heparin along the clinical pipeline. We have determ...

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Détails bibliographiques
Publié dans:Pharmaceutics
Auteurs principaux: Lantero, Elena, Aláez-Versón, Carlos Raúl, Romero, Pilar, Sierra, Teresa, Fernàndez-Busquets, Xavier
Format: Artigo
Langue:Inglês
Publié: MDPI 2020
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7557421/
https://ncbi.nlm.nih.gov/pubmed/32872434
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics12090825
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