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Safety, pharmacokinetics, and pharmacodynamics of Gln‐1062, a prodrug of galantamine

INTRODUCTION: Gln‐1062 (MEMOGAIN) is an intranasally administered lipophilic prodrug of galantamine. Based on high brain‐to‐blood concentrations observed in pre‐clinical studies, Gln‐1062 is expected to have superior cognitive efficacy compared to oral galantamine. METHODS: Forty‐eight healthy elder...

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Publicat a:Alzheimers Dement (N Y)
Autors principals: Bakker, Charlotte, van der Aart, Jasper, Hart, Ellen P., Klaassen, Erica S., Bergmann, Kirsten R., van Esdonk, Michiel J., Kay, Denis G., Groeneveld, Geert Jan
Format: Artigo
Idioma:Inglês
Publicat: John Wiley and Sons Inc. 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7551138/
https://ncbi.nlm.nih.gov/pubmed/33083515
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/trc2.12093
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